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PHARMACEUTICAL FORMULATIONS OF TROPOMYOSIN RELATED KINASE (TRK) INHIBITORS
专利权人:
发明人:
LIEBERMAN HARVEY,YANG DONGLAI,PHILBROOK C MICHAEL,SANTOS MICHAEL,HO CHRIS
申请号:
IN201737025475
公开号:
IN201737025475A
申请日:
2017.07.18
申请国别(地区):
IN
年份:
2017
代理人:
摘要:
Pharmaceutical formulations with a tropomyosin related kinase inhibitor (Trk inhibitor) are disclosed. The pharmaceutical formulations comprise 3 (3 methoxy 4 ((4 methoxybenzyl)oxy)benzyl) 6 (1 methyl 1H pyrazol 4 yl) 3H imidazo[4 5 b]pyridin 2 amine in microcrystalline suspension formulations in its monohydrate form which shows improved characteristics over the anhydrate form and in extended release formulations. The extended release pharmaceutical formulations comprise 3 (3 methoxy 4 ((4 methoxybenzyl)oxy)benzyl) 6 (1 methyl 1H pyrazol 4 yl) 3H imidazo[4 5 b]pyridin 2 amine loaded microspheres.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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