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1,5-dihydro-4h-pyrazolo [3,4-d] pyrimidin-4-ones and 1,5-dihydro-4h-pyrazolo [4,3-c] pyridin-4-ones as inhibitors of pde1
专利权人:
H. LUNDBECK A/S
发明人:
JAN KEHLER,KARSTEN JUHL,LARS KYHN RASMUSSEN,MAURO MARIGO,MIKKEL JESSING,MORTEN LANGGÅRD,PAULO JORGE VIEIRA VITAL
申请号:
BR112017026278
公开号:
BR112017026278A2
申请日:
2017.04.07
申请国别(地区):
BR
年份:
2018
代理人:
摘要:
the present invention provides 1,5-dihydro-4h-pyrazolo [3,4-d] pyrimidin-4-ones and 1,5-dihydro-4h-pyrazolo [4,3-c] pyridin-4-one of formula (i) as inhibitors of pde1 and their use as a medicament, in particular for the treatment of neurodegenerative disorders and psychiatric disorders.a presente invenção proporciona 1,5-di-hidro-4h-pirazolo[3,4-d]pirimidin-4-onas e 1,5-di-hidro-4h-pirazolo[4,3-c]piridin-4-onas da fórmula (i) como inibidores de pde1 e seu uso como um medicamento, em particular para o tratamento de distúrbios neurodegenerativos e distúrbios psiquiátricos.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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