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Process for producing bicycloaniline derivatives
专利权人:
Shuntaro Furukawa
发明人:
Shuntaro Furukawa,Taketo Ikeno,Shinji Kato,Masashi Kawasaki,Hisaki Kojima,Wataru Minagawa,Naotaka Sawada,Fuyuki Yamamoto,Sachin Lohani,Yaling Wang
申请号:
US12996801
公开号:
US08507504B2
申请日:
2009.06.02
申请国别(地区):
US
年份:
2013
代理人:
摘要:
The present invention relates to a process for producing a hydrate of 3-(2,6-dichlorophenyl)-4-imino-7-[(2′-methyl-2′,3′-dihydro-1′H-spiro[cyclopropane-1,4′-isoquinolin]-7′-yl)amino]-3,4-dihydropyrimido[4,5-d]pyrimidin-2(1H)-one (Compound A) or of a pharmaceutically acceptable salt of Compound A and a crystalline form of Compound A or of a pharmaceutically acceptable salt of Compound A, which are useful in the field of treatment of various cancers as a kinase inhibitor, especially as a Weel kinase inhibitor.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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