您的位置: 首页 > 农业专利 > 详情页

Benzimidazole inhibitors of respiratory syncytial virus
专利权人:
JANSSEN R&D IRELAND
发明人:
申请号:
ARP110104739
公开号:
AR085203A1
申请日:
2011.12.16
申请国别(地区):
AR
年份:
2013
代理人:
摘要:
Benzene, which inhibits RSV replication, contains these compounds as active ingredients, and the process for preparing these compounds and compounds. Claim 1: compound (1) represented by formula,a. Prof, N-O x, additional Sal, quarterlia amine, metal complex, or an isomer according to its stereochemical form, wherein each x is independent of C or N; R1 is h; R2 is selected from BR and Cl groups; R3 is - (cr8310; r8311); - r834512;R83088 was selected from group H, cycloquilo c832318327a;alquenilo C- (CR R) -R-Ch832222-p-fluoroofeney, ch8322; (CF) 83323y-so8322; (ch832323);R⁵ is present where X is C, whereby each R⁵ is selected, each independently, from the group consisting of H, C₁₋₆ alkyl,C₁₋₆ alkoxy,halogen, and CN; R⁵ is absent when X is N; R⁶ and R⁷ are each independently chosen from H and C₁₋₁₀ alkyl,C₃₋₇ cycloalkyl,O r8310a and r8311a are added together to form a crystal or aromatic ring of 5 to 6 members, optionally including one or more heteroatoms selected from group n, s and O; r831222 is selected from group H, oh, CF 2323;CHF83222,F Cl SO CHSO₂-C₃₋₇ cycloalkyl,8310; 18322; 8310;R8322; No. 8310; r8311;NR⁶SO₂-C₃₋₇ cycloalkyl,Cn, No. 8310; r8311;COOH, COOR⁶,CONR ROCO-C₁₋₆ alkyl,CONR SO RCONHR SO RCONHR SO NR R CONR SO NR RDibenzoyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldiacyldi.Bencimidazoles que tienen actividad inhibidora sobre la replicación de RSV, composiciones que contienen estos compuestos como ingrediente activo y procesos para preparar estos compuestos y composiciones. Reivindicación 1: Un compuesto representado por la fórmula (1), un profármaco, N-óxido, sal de adición, amina cuaternaria, complejo metálico, o una forma isómerica según la estereoquímica del mismo;
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
相关发明人
相关专利

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充