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2. The process of preparing Jak1 inhibitor (Application Department 1790-2018);
专利权人:
INCYTE CORPORATION
发明人:
LIU PINGLI,WANG DENGJIN,WU YONGZHONG,XIA MICHAEL,ZHOU JIACHENG,CHEN SHILI,JIA ZHONGJIANG,QIAO LEI,FRIETZE WILLIAM,DAI YINGRUI
申请号:
CL2019002032
公开号:
CL2019002032A1
申请日:
2019.07.19
申请国别(地区):
CL
年份:
2019
代理人:
摘要:
The preparation process of F amp compound; oacute; rmula II, including the termination of a 2 - (2R, 5S) - 5 - (2 - ((R) - 1-hydroxy) - 1H imidazo [4, 5-d] tieno [3],2-B] pyridine-1-tetrahydro-2h-piran-2-il) acrylonitrile in a solvent element including water or separation of F amp compounds; oacute; rmula II, the first mixture including 2 - (2R, 5S) - 5 - (2 - ((R) - 1-hydroxy) - 1 h-pyridan [4, 5-d] tieno [3], 2-B] pyridine-1-il (tetrahydro-2h-piran-2-il) acetone and solvent components, including isopropanol and water; / P gt;<;p>;UN PROCESO PARA PREPARAR UN COMPUESTO DE FÓ;RMULA II, QUE COMPRENDE SUSPENDER UNA FORMA ANHIDRA DE 2-((2R,5S)-5-(2-((R)-1-HIDROXIETIL)-1H-IMIDAZO[4 ,5-D]TIENO[3 , 2-B]PIRIDIN-1 -TETRAHIDRO-2H-PIRAN-2-IL)ACETONITRILO EN UN COMPONENTE SOLVENTE QUE COMPRENDE AGUA O QUE COMPRENDE AISLAR EL COMPUESTO DE FÓ;RMULA II DE UNA PRIMERA MEZCLA QUE COMPRENDE 2-((2R,5S)-5-(2-((R)-1 -HIDROXIETIL)-1 H-IMIDAZO[4,5-D]TIENO[3,2-B]PIRIDIN-1 - IL)TETRAHIDRO-2H-PIRAN-2-IL)ACETONITRILO Y UN COMPONENTE SOLVENTE QUE COMPRENDE ISOPROPANOL Y AGUA.<;/p>;
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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