A dual targeting drug carrier is provided. The dual targeting drug carrier comprises a first targeting molecule and a second targeting molecule, wherein the targeting molecule comprises peptide, antibody, or protein. The targeting molecule can be bound to specific receptors, proteins, or glycoproteins to recognize the specific tumor cells, tissues, or organs. The dual targeting drug carriers are further conjugated with imaging agents, radioactive molecules (radiopharmaceuticals, isotopes, or chemotherapeutic drugs) or nanoparticles to form a conjugate.本發明係提供一雙重標靶藥物載體,包括一第一標靶分子以及一第二標靶分子,其中標靶分子包括胜肽、抗體或蛋白質。本發明之標靶分子可結合至特定的受體、特異性蛋白或醣蛋白等,以辨識特定腫瘤細胞、組織或器官。本發明之雙重靶分子更可與一成像物質、放療物質(放射性藥物、同位素或化療藥物)或奈米顆粒共軛結合,形成一共軛物。