您的位置: 首页 > 农业专利 > 详情页

INHIBITEUR DE CASÉINE KINASE 1DELTA ET CASÉINE KINASE EPSILON
专利权人:
PHARMADESIGN, INC.;NB HEALTH LABORATORY CO. LTD.
发明人:
申请号:
EP11816390.6
公开号:
EP2604606B1
申请日:
2011.08.08
申请国别(地区):
EP
年份:
2014
代理人:
摘要:
There is provided a novel oxazolone derivative having inhibitory activity against casein kinase 1´ and casein kinase 1µ. In addition, the present inhibitor inhibits casein kinase 1´ and casein kinase 1µ, and thus there is also provided a pharmaceutical agent useful for the treatment and/or prevention of diseases, with the pathological conditions of which the activation mechanism of casein kinase 1´ or casein kinase 1µ is associated. There is further provided a pharmaceutical agent useful for the treatment of, particularly, circadian rhythm disorder (including sleep disorder), central neurodegenerative disease, and cancer. An inhibitor of casein kinase 1´ and casein kinase 1µ comprising, as an active ingredient, an oxazolone derivative represented by the following general formula (1), a salt thereof, a solvate thereof, or a hydrate thereof: wherein X represents a halogen atom (which may be any one of a fluorine atom, a chlorine atom, a bromine atom, and an iodine atom).
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充