EIS, Knut,PÜHLER, Florian,ZORN, Ludwig,SCHOLZ, Arne,LIENAU, Philip,GNOTH, Mark Jean,BÖMER, Ulf,GÜNTHER, Judith,FANGHÄNEL, Jörg,KORR, Daniel
申请号：
ES12729041
公开号：
ES2625854T3
申请日:
2012.05.30
申请国别(地区):
ES
年份:
2017
代理人:
摘要：
A compound of general formula (I): ** Formula ** in which: A represents a group selected from: ** Formula ** in which one or more R3 substituents, independent of one another, is present (s) ) in any position of group A； and in which * indicates the point of union of said groups with the rest of the molecule； R1 represents a C1-C6 alkyl group, said group being substituted with one or more -OH groups and optionally substituted with one or more substituents independently selected from: a halogen atom, a -CN group, C1-C6 alkyl, C2 alkenyl C6, C2-C6 alkynyl, C3-C10 cycloalkyl, 3-10 membered heterocycloalkyl, aryl, aryl substituted with one or more substituents R, heteroaryl, - C (>； = O) R ', -C (>； = O) NH2 , -C (>； = O) N (H) R ', - C (>； = O) N (R') R ", -C (>； = O) OR ', -NH2, -NHR', -N ( R ') R ", -N (H) C (>； = O) H, - N (H) C (>； = O) R', -N (R ') C (>； = O) H, -N ( R ') C (>； = O) R', -N (H) C (>； = O) NH2, -N (H) C (>； = O) NHR ', -N (H) C (>； = O) N (R ') R ", - N (R') C (>； = O) NH2, -N (R ') C (>； = O) NHR', -N (R ') C (>； = O) N (R ') R ", -N (H) C (>； = O) OR', - N (R ') C (>； = O) OR', -N (H) S (>； = O) R ', - N (R ') S (>； = O) R', -N (H) S (>； = O) NH2, -N (H) S (>； = O) NHR ', - N (H) S (>； = O) N (R ') R ", -N (R') S (>； = O) NH2, -N (R ') S (>； = O) NHR', - N (R ') S (>； = O) N (R ') R ", -N (H) S (>； = O) 2R', -N (R ') S (>； = O) 2R', -N>； = S (>； = O) ( R ') R ", -OH, C1-C6 alkoxy, -OC (>； = O) R', - OC (>； = O) NH2, -OC (>； = O) NHR ', -OC (>； = O) N (R ') R ", -SH, C1-C6-S alkyl, -S (>； = O) 2NH2, - S (>； = O) 2NHR ', - S (>； = O) 2N (R') R ", -S (>； = O) (>； = NR ') R", -S (>； = O) R ', -S (>； = O) 2R'； R2 represents a C1-C6 alkyl group or a C3-C10 cycloalkyl group, in which C1-C6 alkyl, or C3-C10 cycloalkyl is optionally substituted one or more times with a substituent selected from: - Hal, or a -OH group , C1-C6 alkoxy, C1-C6 haloalkoxy； R3 represents a substituent
