ALAN PETERSON GRAVES III,JAMES A. BRACKLEY III,KENNETH ALLEN NEWLANDER,KENNETH C. MCNULTY,STEVEN DAVID KNIGHT,XINRONG TIAN
申请号:
BR112017028616
公开号:
BR112017028616A2
申请日:
2016.06.30
申请国别(地区):
BR
年份:
2018
代理人:
摘要:
The present invention relates to novel compounds according to formula (I) which are inhibitors of zest homologue enhancer 2 (ezh2), pharmaceutical compositions containing them, processes for their preparation, and their use in therapy. for the treatment of cancers.a presente invenção refere-se a compostos inovadores de acordo com a fórmula (i) que são inibidores de acentuador de homólogo de zeste 2 (ezh2), a composições farmacêuticas contendo os mesmos, a processos para sua preparação, e a seu uso na terapia para o tratamento de cânceres.