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Antiretroviral Complexes and Their Use (ADC)
专利权人:
ABBVIE INC.
发明人:
REILLY, EDWARD B.,ANDERSON, MARK
申请号:
ARP180100866
公开号:
AR111363A1
申请日:
2018.04.06
申请国别(地区):
AR
年份:
2019
代理人:
摘要:
Claim 1: A set of antibodies (ADC) containing the (1) structure,Or salt, where AB includes an anti-PRLR antibody, including: (1) a heavy chain variable region, including a CDR1 sequence, including SEQ ID No.3, a CDR2 sequence, including SEQ ID No.4, and a CDRH3 Qua sequence, including SEQ ID No.4. 5. (2) A region of light chain variables, including CDR1 sequence No. 8 of Chemical Abstracts, CDR2 sequence No. 9 of Chemical Abstracts and CDR3 sequence No. 10 of Chemical Abstracts, and a variation of S239C in a continuous P-chain region. A. ESADA, numbered in accordance with KABAT;(4) N is about 2. Claim 12: A synthetic antibody (ADC) containing (2) formula structure,Or salt, where D includes a pyrethroid (PBD);AB is an anti-acrylic receptor antibody.This is Val, Z is Ala, Q is 1, 2, 3, 4, 5, 6, 7, or 8. Anti-PRLR antibodies include: (1) a heavy chain variable region, including a CDR1 sequence, including SEQ ID No. 3, a CDR2 sequence, including SEQ ID No. 4, and a purchased CDR3 sequence. (2) A light chain variable region, including CDR1 sequence, including SEQ ID No.8, CDR2 sequence, including SEQ ID No.9 and CDR3 sequence, including SEQ ID No.10; and (3) variation of S239C included in CONS region. A. Heavy chain test, whose number is in accordance with KABAT;(4) N is about 2.Reivindicación 1: Un conjugado de anticuerpo-fármaco (ADC) que comprende la estructura de la fórmula (1), o una sal del mismo, en el que Ab comprende un anticuerpo anti-PRLR que comprende: i) una región variable de cadena pesada que comprende una secuencia de CDRH1 que comprende la SEQ ID Nº 3, una secuencia de CDRH2 que comprende la SEQ ID Nº 4, y una secuencia de CDRH3 qua comprende la SEQ ID Nº 5; ii) una región variable de cadena ligera que comprende una secuencia de CDRL1 que comprende la SEQ ID Nº 8, una secuencia de CDRL2 que comprende la SEQ ID Nº 9, y una secuencia de CDRL3 que comprende la SEQ ID Nº 10; iii) una mutación que comprende S239C en una región constante de cadena pesada, en l
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