System of the present invention provides a series of novel 1, the disubstituted vinegar amido anthraquinone derivative of 2-, and further provide for the preparation method and applications of those derivatives, the application is comprising using the analog derivative as the medical composition for the treatment of cancer, and its application has the growth of poisoning tumour cell, cancer cell, and then treating cancer and other effects comprising the analog derivative.本發明係提供一系列新穎1,2-雙取代醯胺基蒽醌衍生物，並進一步提供該些衍生物之製備方法及其應用，該應用包含將該類衍生物作為治療癌症之醫藥組合物，且其應用包含該類衍生物具有毒殺腫瘤細胞、癌細胞之生長，進而治療癌症等功效。
