您的位置: 首页 > 农业专利 > 详情页

DERIVE DE 2-ACYLAMINOTHIAZOLE OU SEL DE CELUI-CI
专利权人:
ASTELLAS PHARMA INC.
发明人:
TAKAHASHI, TAISUKE,KOIKE, TAKANORI,NEGORO, KENJI,TANAKA, HIROAKI,MAEDA, JUN,YOKOYAMA, KAZUHIRO,TAKAMATSU, HAJIME
申请号:
CA2950564
公开号:
CA2950564A1
申请日:
2015.06.05
申请国别(地区):
CA
年份:
2015
代理人:
摘要:
[Problem] To provide a compound useful as an active ingredient of a pharmacological composition for the treatment of urinary storage symptoms, dysuria, lower urinary tract diseases, and the like. [Solution] The inventors perfected the present invention after discovering that thiazole derivatives substituted at position 2 by pyrazinylcarbonylamino are exceptional muscarinic M3 receptor positive allosteric modulators and can be expected to serve as agents for the prevention or treatment of urinary bladder and urinary tract diseases involving bladder contraction mediated by muscarinic M3 receptors. The 2-acylaminothiazole derivatives or salts thereof of the present invention can be expected to serve as agents for the prevention or treatment of urinary bladder and urinary tract diseases involving bladder contraction mediated by muscarinic M3 receptors, e.g., underactive bladder and the like.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充