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aqueous suspension, injectable preparation, and filled syringe
专利权人:
LTD.;OTSUKA PHARMACEUTICAL CO.
发明人:
Hidekazu Toyofuku,Takuya Minowa,Tetsuya Sato,YUSUKE HOSHIKA
申请号:
BR112014026398
公开号:
BR112014026398A2
申请日:
2013.04.23
申请国别(地区):
BR
年份:
2017
代理人:
摘要:
1/1 Summary "Aqueous suspension, injectable preparation, and filled syringe" The present invention addresses the problem of providing an injectable release formulation. release to a therapeutically effective amount of 7- [4- (4-benzo [b] thiophen-4-yl-piperazin-1-yl) butoxy] -1h-quinolin-2-one for at least one week as a long action form of the medication administration for 7- [4- (4-benzo [b] thiophen-4-yl-piperazin-1-yl) butoxy] -1h -quinolin-2-one. The present invention provides an injectable preparation at the concentration of which in the blood can be maintained for at least one week, the formulation comprising 7- [4- ( 4-benzo [b] thiophen-4-yl-piperazin-1-yl) butoxy] -1h-quinolin-2-one or a salt thereof as an active ingredient.1 / 1 resumo “suspensãƒo aquosa, preparaã‡ãƒo injetã�vel, e, seringa preenchidaâ€� a presente invenã§ã£o trata o problema do fornecimento de uma formulaã§ã£o injetã¡vel de liberaã§ã£o prolongada para liberar uma quantidade terapeuticamente eficaz de 7-[4-(4-benzo[b]tiofen-4-il-piperazin-1-il)butã³xi]- 1h-quinolin-2-ona por pelo menos uma semana, como uma forma de aã§ã£o longa da administraã§ã£o de medicaã§ã£o para a 7-[4-(4-benzo[b]tiofen-4-il- piperazin-1-il)butã³xi]-1h-quinolin-2-ona. a presente invenã§ã£o fornece uma preparaã§ã£o injetã¡vel a concentraã§ã£o da qual no sangue pode ser mantida por pelo menos uma semana, a formulaã§ã£o compreendendo a 7-[4-(4- benzo[b]tiofen-4-il-piperazin-1-il)butã³xi]-1h-quinolin-2-ona ou um sal da mesma como um ingrediente ativo.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
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