您的位置: 首页 > 农业专利 > 详情页

substituted oxazolidinones, process for their production, use thereof and process for preventing in vitro blood coagulation.
专利权人:
发明人:
ALEXANDER STRAUB,THOMAS LAMPE,JENS POHLMANN,SUSANNE ROEHRIG,ELISABETH PERZBORN,KARL-HEINS SCHLEMMER,JOSEPH PERNERSTORFER
申请号:
BR0017050
公开号:
BR0017050B1
申请日:
2000.12.11
申请国别(地区):
BR
年份:
2012
代理人:
摘要:
N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides (I) and their salts, hydrates and prodrugs are new. N-oxazolidinylmethyl-substituted (benzo)thiophene carboxamides of formula (I) and their salts, hydrates and prodrugs are new. [Image] R 1>; : optionally benzo-fused thiophene, optionally substituted one or more times; R 2>; : any selected organic group; R 3>;-R 8>; : same or different hydrogen or 1-6C alkyl. Excluded are compounds where R 2>; = phenyl (optionally substituted once or more) and all of R 3>;-R 8>; are hydrogen. Independent claims are also included for the following: (1) preparation of (I); and (2) pharmaceutical composition containing (I), optionally also auxiliaries and carriers. ACTIVITY : Anticoagulant; cardiant; anti-anginal; vasotropic; thrombolytic; cerebroprotective; antiarthritic; antiarteriosclerotic; cytostatic; nootropic; neuroprotective. Test details are described but no results given. MECHANISM OF ACTION : Coagulation factor Xa Inhibitor.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充