BERGER, RICHARD A.,伯格 理查A,伯格 理查A,HOFFMANN, CHRISTIAN,渥夫曼 克里斯汀,渥夫曼 克里斯汀,MARSHALL, WILLIAM J.,马雪尔 威廉J,馬雪爾 威廉J,SHAPIRO, RAFAEL,雪彼罗 瑞发艾,雪彼羅 瑞發艾
申请号：
TW101133631
公开号：
TWI577286B
申请日:
2012.09.14
申请国别(地区):
TW
年份:
2017
代理人:
摘要：
Disclosed are solid forms of 8-chloro-N-[(2-chloro-5-methoxyphenyl)sulfonyl]-6-(trifluoromethyl)-imidazo[1,2-a]pyridine-2-carboxamide (Compound 1). Methods for the preparation of solid forms of Compound 1 and for the conversion of one solid form of Compound 1 into another are disclosed.Disclosed are nematocidal compositions comprising a nematocidally effective amount of a solid form of Compound 1 and at least one additional component selected from the group consisting of surfactants, solid diluents and liquid carriers. Compositions comprising a mixture of a solid form of Compound 1 and at least one other nematicide, insecticide and/or fungicide are also disclosed.Also disclosed are methods for protecting a plant from nematodes comprising applying to the plant, or portion, or seed thereof, or to the growing medium of the plant, a nematocidally effective amount of Compound 1 comprising the polymorph Form A.本發明係揭露8-氯-N-[(2-氯-5-甲氧苯基)磺醯基]-6-(三氟甲基)-咪唑[1,2-a]吡啶-2-甲醯胺(化合物1)之固體形態。本發明並提供製備化合物1固體形態及將化合物1之一種固體形態轉換為另一種固體形態的方法。本發明揭露殺線蟲組成物,其包含殺線蟲有效量之化合物1之固體形態及至少一種選自於由界面活性劑、固體稀釋劑以及載液所組成之群組的額外成分。亦揭露包含化合物1之固體形態及至少一種其他殺線蟲劑、殺蟲劑及/或殺真菌劑之混合物的組成物。本發明亦揭露保護植物免受線蟲侵害之方法,包含施用一殺線蟲有效量之包括多形體形態A之化合物1至該植物或其部分或種子或至該植物的生長介質。
