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NEW BENZODIOXOLPIPERIDINES
专利权人:
Ф. ХОФФМАНН-ЛЯ РОШ АГ (CH)
发明人:
РОДРИГЕЗ САРМИЕНТО Роза Мария (CH),ВИХМАНН Юрген (DE)
申请号:
RU2013142013/04
公开号:
RU2013142013A
申请日:
2012.02.29
申请国别(地区):
RU
年份:
2015
代理人:
摘要:
1. Compounds having the formula (I) in which n is 0, 1, 2 or 3; Y is —C (O) - or —S (O) -; R is a hydrogen atom, a halogen atom, cyano, alkyl, haloalkyl, hydroxy, alkoxy, haloalkoxy, cycloalkyl, heterocycloalkyl, aryl, heteroaryl, -NRR, -C (O) -NRR or -S (O) -R; moreover, alkyl, haloalkyl and alkoxy are optionally substituted with one, two or three independent R groups; and cycloalkyl, heterocycloalkyl, aryl and heteroaryl are optionally substituted with one, two or three independent R groups; R, R, R independently represent a hydrogen atom, a halogen atom, cyano, alkyl, haloalkyl, hydroxy, alkoxy or haloalkoxy; R represents cyano, hydroxy, alkoxy, cycloalkyl, heterocycloalkyl, aryl or heteroaryl, moreover, cycloalkyl, heterocycloalkyl, aryl and heteroaryl are optionally substituted with one, two or three independent R groups; R represents a halogen atom, cyano, alkyl, haloalkyl, hydro and, alkoxy, haloalkoxy, oxo, cycloalkyl, heterocycloalkyl, aryl or heteroaryl; R, independently represent a hydrogen atom, alkyl, cycloalkyl, cycloalkylalkyl, heterocycloalkyl, heterocycloalkylalkyl, aryl or heteroaryl; moreover, cycloalkyl, heterocycloalkyl, aryl and heteroaryl are optionally substituted with one, two or three independent R groups; R is alkyl, cycloalkyl, heterocycloalkyl, aryl, heteroaryl or —NRR; moreover, cycloalkyl, heterocycloalkyl, aryl and heteroaryl are optionally substituted with one, two or three independent R groups; R represents a halogen atom, cyano, alkyl, haloalkyl, hydroxy, alkoxy, haloalkoxy or oxo; R represents a halogen atom, cy1. Соединения, имеющие формулу (I),в которыхn равно 0, 1, 2 или 3;Y представляет собой -С(О)- или -S(O)-;Rпредставляет собой атом водорода, атом галогена, циано, алкил, галогеноалкил, гидрокси, алкокси, галогеноалкокси, циклоалкил, гетероциклоалкил, арил, гетероарил, -NRR, -C(O)-NRRили -S(O)-R; причем, алкил, галогеноалкил и алкокси необязательно замещены одной, двумя или тремя независимыми группами R; и циклоалкил, гетероц
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
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