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Inhibitors myristate small molecules BCR-ABL and methods of use
- 专利权人:
- Inc.;Dana-Farber Cancer Institute;Dana-Farber Cancer Institute, Inc.;The Scripps Research Institute
- 发明人:
- GRAY, Nathanael,ZHANG, Jianming,OKRAM, Barun,DENG, Xianming,CHANG, Jae Won,WOJCIECHOWSKI, Amy
- 申请号:
- ES08857261
- 公开号:
- ES2610190T3
- 申请日:
- 2008.11.28
- 申请国别(地区):
- ES
- 年份:
- 2017
- 代理人:
- 摘要:
- A compound selected from the following: 4- (6- (4- (trifluoromethoxy) phenylamino) -5-methyl-pyrimidin-4-yl) -N- (2-morpholinoethyl) benzamide; 6- (1H-pyrrolo [2,3-b] pyridin-1-yl) -N- (4- (trifluoromethoxy) phenyl) pyrimidin-4-amine; N- (4- (trifluoromethoxy) phenyl) -6- (1,3,5-trimethyl-1H-pyrazol-4-yl) pyrimidin-4-amine; 4- [5-Methyl-6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] benzenesulfonamide; N-Methyl-4- [5-methyl-6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] benzenesulfonamide; N-Ethyl-4- [6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] benzenesulfonamide; N- (2-Hydroxy-ethyl) -4- [6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] benzenesulfonamide; [6- (4-Methanesulfonyl-phenyl) -pyrimidin-4-yl] - (4-trifluoromethoxy-phenyl) -amine; [6- (4-Methanesulfonyl-phenyl) -5-methyl-pyrimidin-4-yl] - (4-trifluoromethoxyphenyl) -amine; {6- [4- (propane-2-sulfonyl) -phenyl] -pyrimidin-4-yl} - (4-trifluoromethoxy-phenyl) -amine; {5-Methyl-6- [4- (propane-2-sulfonyl) -phenyl] -pyrimidin-4-yl} - (4-trifluoromethoxy-phenyl) -amine; N, N-Diethyl-4- [6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] benzenesulfonamide; N, N-Diethyl-4- [5-methyl-6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] -benzenesulfonamide; {6- [4- (Piperidine-1-sulfonyl) -phenyl] -pyrimidin-4-yl} - (4-trifluoromethoxy-phenyl) -amine; 4-Methyl-N- {4- [6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] -phenyl} -benzenesulfonamide; 4-Methyl-N- {4- [5-methyl-6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] -phenyl} -benzenesulfonamide; N- {4- [6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] -phenyl} -methanesulfonamide; {4- [6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] -phenyl} -amide; {4- [6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] -phenyl} butane-1-sulfonic acid; {4- [6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] -phenyl} propane-2-sulfonic acid; {4- [6- (4-trifluoromethoxy-phenylamino) -pyrimidin-4-yl] -phenyl} pentane-2-sulfonic acid
- 来源网站:
- 中国工程科技知识中心
- 来源网址:
- http://www.ckcest.cn/home/