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DERIVATIVES OF N - [(1H-PYRAZOL-1-YL) ARYL] - 1H - INDOLE OR 1H – INDAZOLE - 3 - CARBOXAMIDE, THEIR PREPARATION AND THEIR USE AS P2Y12 ANTAGONISTS
专利权人:
SANOFI
发明人:
BADORC ALAIN,BOLDRON, CHRISTOPHE,DELESQUE, NATHALIE,FOSSEY, VALÉRIE,LASSALLE, GILBERT,YVON, XAVIER
申请号:
MYPI 2013003927
公开号:
MY161202A
申请日:
2011.09.13
申请国别(地区):
MY
年份:
2017
代理人:
摘要:
THE PRESENT INVENTION RELATES TO COMPOUNDS CORRESPONDING TO FORMULA (I): IN WHICH: - A REPRESENTS A DIVALENT AROMATIC RADICAL; - X REPRESENTS A -CH- GROUP OR A NITROGEN ATOM; - R1 REPRESENTS A (C1-C4) ALKYL OR A (C1-C4) ALKOXY; - R2 REPRESENTS A GROUP ALK; - R3 REPRESENTS A HYDROXYL OR A GROUP -NR7R8; - R4 REPRESENTS A HYDROGEN ATOM, A HALOGEN ATOM, A CYANO, A PHENYL, A GROUP ALK, A GROUP OALK OR A GROUP -NR9R10; - R5 REPRESENTS A HYDROGEN ATOM, A HALOGEN ATOM OR A GROUP ALK; - R6 REPRESENTS A HYDROGEN ATOM, A HALOGEN ATOM, A CYANO, A GROUP -COOALK OR A -CONH2 GROUP; AND METHOD OF PREPARATION AND APPLICATION IN THERAPEUTICS.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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