COMBS, ANDREW P.,DOUTY, BRENT,GLENN, JOSEPH,HE, CHUNHONG,LI, YUN-LONG,ZHU, WENYU,MEI, SONG,SPARKS, RICHARD B.,YAO, WENQING,YUE, EDDY W.,MADUSKUIE JR., THOMAS P.
申请号:
PE2015001833
公开号:
PE20151996A1
申请日:
2014.02.28
申请国别(地区):
PE
年份:
2016
代理人:
摘要:
The application provides a method for treating disorders related to PI3K (delta) by using a formula compound, or a drug acceptable salt using a formula compound, wherein R2 is C1-C6 tar, etc.; R4 is halogen, oh, etc.; R5 is halogen, oh, etc.; CY is cyclo c3-7. The diseases to be treated include pure specific hemoglobin, autoimmune anemia, vasculitis and so on.La presente solicitud proporciona metodos para tratar trastornos relacionados con PI3K(delta) utilizando compuestos de la formula I, o sales farmaceuticamente aceptables de los mismos, donde R2 es alquilo C1-C6, etc.; R4 es halo, OH, etc.; R5 es halo, OH, etc.; Cy es cicloalquilo C3-7, etc. Las enfermedades a tratar son purpura trombocitopenica idiopatica, anemia hemolitica autoinmune, vasculitis, etc