您的位置: 首页 > 农业专利 > 详情页

highly water soluble salts of a short acting phenylalkylamine calcium channel blocker and uses thereof
专利权人:
MILESTONE PHARMACEUTICALS INC.
发明人:
MARTIN P. MAGUIRE
申请号:
BR112017021620
公开号:
BR112017021620A2
申请日:
2016.04.13
申请国别(地区):
BR
年份:
2018
代理人:
摘要:
The present invention surprisingly includes water-soluble salts of a phenylalkylamine compound which are potent type 1 calcium channel antagonists. Aqueous solutions including the salts of the present invention are formulated for nasal administration and provide a novel therapeutic platform for the treatment of stable angina, migraine and cardiac arrhythmia, such as paroxysmal supraventicular tachycardia.a presente invenção inclui surpreendentemente sais solúveis em água de um composto de fenilalquilamina que são antagonistas potentes de canais de cálcio do tipo l. as soluções aquosas que incluem os sais da presente invenção são formuladas para administração nasal e fornecem uma nova plataforma terapêutica para o tratamento de angina estável, enxaqueca e arritmia cardíaca, tal como taquicardia supraventicular paroxismal.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充