Anthony BEAUGLEHOLE;Robert D. THOMPSON;Jayson M. RIEGER
发明人:
Anthony BEAUGLEHOLE,Jayson M. RIEGER,Robert D. THOMPSON
申请号:
US13190136
公开号:
US20120035192A1
申请日:
2011.07.25
申请国别(地区):
US
年份:
2012
代理人:
摘要:
The present invention provides compounds of formulae Ia and Ib:wherein R1-5, Q, X, Y, Z, p, q, and r are as defined herein. The compounds are potent and selective antagonists of A2A adenosine receptors (ARs). The invention further includes pharmaceutical compositions containing these compounds and methods of using the same.