Derivati 5-(2-(piridin-2-ilamino)-1,3-tiazol-5-il)-2,3-dihidro-1H-izoindol-1- ona in njihova uporaba kot dvojni inhibitorji fosfatidilinozitol 3- kinaze delta in gama
PERRY Matthew,KARABELAS Konstantinos,MOGEMARK Mickael,BOLD Peter,TYRCHAN Christian,NIKITIDIS Antonios,PETERSEN Jens,BORJESSON Ulf
申请号:
SI201730357
公开号:
SI3515910T1
申请日:
2017.09.21
申请国别(地区):
SI
年份:
2020
代理人:
摘要:
that inhibit phosphatidylinositol 3-kinase gamma (PI3Kγ) and phosphatidylinositol 3-kinase gamma (PI3Kγ) activity, to their utility in treating and/or preventing clinical conditions including respiratory diseases, such as asthma and chronic obstructive pulmonary disease (COPD), to their use in therapy, to pharmaceutical compositions containing them and to processes for preparing such compounds.