David Edwin THURSTON,Khondaker Mirazur RAHMAN,Shirin JAMSHIDI,Kazi Sharmin NAHAR
申请号：
US16638041
公开号：
US20200216432A1
申请日:
2018.08.10
申请国别(地区):
US
年份:
2020
代理人:
摘要：
The invention relates to novel derivatives of formula (I)where R1, R2, R3, R4, R5, X and m are as defined in the specification. These compounds which have therapeutic activity, in particular, as STAT3 inhibitors and so are useful in the treatment of proliferative diseases or conditions such as cancer. Methods for producing these compounds, novel intermediates used in the methods, pharmaceutical compositions containing them and their use in therapy form further aspects of the invention.
