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compounds, process for their manufacture, method for treating and / or preventing diseases that are modulated by hm74a agonists and uses of the compounds
专利权人:
F. HOFFMANN-LA ROCHE AG
发明人:
AURELIA CONTE,HENRIETTA DEHMLOW,UWE GRETHER,NICOLE A. KRATOCHWIL,HOLGER KUEHNE,ROBERT NARQUIZIAN,CONSTANTINOS PANOUSIS,JENS-UWE PETERS,FABIENNE RICKLIN,STEPHAN ROEVER
申请号:
BRPI0711879
公开号:
BRPI0711879A2
申请日:
2007.05.11
申请国别(地区):
BR
年份:
2012
代理人:
摘要:
COMPOUNDS, PROCESS FOR THEIR MANUFACTURE, METHOD FOR THE TREATMENT AND / OR PREVENTION OF DISEASES THAT ARE MODULATED BY HM74A AGONISTS AND USES OF THE COMPOUNDS The invention relates to new pyridopyrimidinone derivatives of formula (I) in which R ^ 1 ^ to R 8, X, Y, men are as defined in the description and the claims, as well as their physiologically acceptable salts and esters. These compounds are HM74A agonists and can be used as drugs.COMPOSTOS, PROCESSO PARA A SUA MANUFATURA, MéTODO PARA O TRATAMENTO E/OU PREVENçãO DE ENFERMIDADES QUE SãO MODULADAS POR AGONISTAS DE HM74A E USOS DOS COMPOSTOS A invenção relaciona-se com novos derivados de piridopirimidinona da fórmula (I) em que R^ 1^ a R^ 8^ , X, Y, m e n são tais como definidos na descrição e nas reivindicações, bem como os seus sais e ésteres fisiologicamente aceitáveis. Estes compostos são agonistas HM74A e podem ser usados como medicamentos.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
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