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TETRA-HYDROIBENZO-1,4-DIAZEPINS REPLACED BY ARILA AND HETEROARYL AND USE OF THE SAME TO BLOCK NOREPINEPHRINE, DOPAMINE AND SEROTONIN RECAPTATION.
专利权人:
AMR TECHNOLOGY INC.;BRISTOL-MYERS SQUIBB COMPANY
发明人:
PETER R. GUZZO,BRUCE F. MOLINO,WENGE CUI,SHUANG LIU,RICHARD E. OLSON
申请号:
BRPI0811204
公开号:
BRPI0811204A2
申请日:
2008.05.08
申请国别(地区):
BR
年份:
2014
代理人:
摘要:
The aryl- and heteroaryl-substituted tetrahydrobenzo-1,4-diazepine derivative compounds of the present invention are represented by formulae 1(A-D) having the following structure: where the substituents X and R1-R8 are as defined herein.
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