Benzodiazepine bromide control inhibitor

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专利权人:

GLAXOSMITHKLINE LLC

发明人:

GOSMINI, ROMAIN LUC MARIE,MIRGUET, OLIVIER

申请号：

PE2012000614

公开号：

PE20121181A1

申请日:

2010.08.06

申请国别(地区):

PE

年份:

2012

代理人:

摘要：

It refers to a formula (I) benzodiazepine derivative, such as 2 - [(4S) - 6 - (4-Chloro-phenyl) - 1-methyl-8 - (methyloxygen) - 4H - [1, 2, 4] - triazole - [4, 3-A] [1, 4] - benzo-dimethyl-4-1] - n-ethyl-acetyl-ethylamine. A pharmacological composition including this compound was also mentioned. This compound inhibits the association between brominated bet and acetyllysine residues.REFERIDA A UN DERIVADO DE BENZODIAZEPINA DE FORMULA (I) TAL COMO 2-[(4S)-6-(4-CLORO-FENIL)-1-METIL-8-(METILOXI)-4H-[1,2,4]-TRIAZOLO-[4,3-a][1,4]-BENZO-DIAZEPIN-4-IL]-N-ETIL-ACETAMIDA. TAMBIEN ESTA REFERIDA A UNA COMPOSICION FARMACEUTICA QUE COMPRENDE DICHO COMPUESTO (I). DICHO COMPUESTO INHIBE EL ENLACE DE LOS BROMODOMINIOS DE LA FAMILIA BET CON LOS RESIDUOS DE LISINA ACETILADA

来源网站：

中国工程科技知识中心

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