NOVEL ANTIFUNGAL 5,6-DIHYDRO-4H-PYRROLO[1,2-a][1,4]-BENZODIAZEPINES AND 6H-PYRROLO[1,2-a][1,4]BENZODIAZEPINES SUBSTITUTED WITH BICYCLIC BENZENE DERIVATIVES
MEERPOEL, LIEVEN,MAES, LOUIS, JULES, ROGER, MARIE,DE WIT, KELLY
申请号：
MYPI 2013002066
公开号：
MY161360A
申请日:
2011.12.19
申请国别(地区):
MY
年份:
2017
代理人:
摘要：
THE PRESENT INVENTION IS CONCERNED WITH NOVEL ANTIFUNGAL 5,6-DIHYDRO-4H-PYRROLO-[1 ,2-A][1,4]BENZODIAZEPINES AND 6H-PYRROLO[1 ,2-A](1,4)BENZODIAZEPINES SUBSTITUTED WITH BICYCLIC BENZENE DERIVATIVES OF FORMULA (I) WHEREIN R1, R2, R3, R4, R5. R6 AND R7 HAVE THE MEANING DEFINED IN THE CLAIMS. THE COMPOUNDS ACCORDING TO THE PRESENT INVENTION ARE ACTIVE MAINLY AGAINST DERMATOPHYTES AND SYSTEMIC FUNGAL INFECTIONS. THE INVENTION FURTHER RELATES TO PROCESSES FOR PREPARING SUCH NOVEL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS COMPRISING SAID COMPOUNDS AS AN ACTIVE INGREDIENT AS WELL AS THE USE OF SAID COMPOUNDS AS A MEDICAMENT. (NO SUITABLE FIGURE)
