Brian K. Albrecht,Steven F. Bellon,Victor S. Gehling,Jean-Christophe Harmange,Yves LeBlanc,Jun Liang,Steven Magnuson,Vicki Tsui,Birong Zhang
申请号:
US14477566
公开号:
US20150065522A1
申请日:
2014.09.04
申请国别(地区):
US
年份:
2015
代理人:
摘要:
The present invention relates to compounds formula (I):and to salts thereof, wherein R1-R4 and A have any of the values defined in the specification, and compositions and uses thereof. The compounds are useful as inhibitors of histone demethylases, such as KDM5. Also included are pharmaceutically acceptable compositions comprising the compounds of the present invention and methods of using said compositions in the treatment of various disorders.