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IMIDAZOLE DERIVATIVES AS PDE10A ENZYME INHIBITORS
专利权人:
H. LUNDBECK A/S
发明人:
KEHLER, JAN,NIELSEN, JACOB,MARIGO, MAURO,KILBURN, JOHN PAUL,LANGGARD, MORTEN
申请号:
MYPI 2013001727
公开号:
MY163327A
申请日:
2011.11.18
申请国别(地区):
MY
年份:
2017
代理人:
摘要:
THIS INVENTION IS DIRECTED TO COMPOUNDS, WHICH ARE PDE10A ENZYME INHIBITORS. THE INVENTION PROVIDES A PHARMACEUTICAL COMPOSITION COMPRISING A THERAPEUTICALLY EFFECTIVE AMOUNT OF A COMPOUND OF THE INVENTION AND A PHARMACEUTICALLY ACCEPTABLE CARDER. THE PRESENT INVENTION ALSO PROVIDES PROCESSES FOR THE PREPARATION OF THE COMPOUNDS OF FORMULA I. THE PRESENT INVENTION FURTHER PROVIDES A METHOD OF TREATING A SUBJECT SUFFERING FROM A NEURODEGENERATIVE DISORDER COMPRISING ADMINISTERING TO THE SUBJECT A THERAPEUTICALLY EFFECTIVE AMOUNT OF A COMPOUND OF FORMULA I. THE PRESENT INVENTION ALSO PROVIDES A METHOD OF TREATING A SUBJECT SUFFERING FROM A DRUG ADDICTION COMPRISING ADMINISTERING TO THE SUBJECT A THERAPEUTICALLY EFFECTIVE AMOUNT OF A COMPOUND OF FORMULA I. THE PRESENT INVENTION FURTHER PROVIDES A METHOD OF TREATING A SUBJECT SUFFERING FROM A PSYCHIATRIC DISORDER COMPRISING ADMINISTERING TO THE SUBJECT A THERAPEUTICALLY EFFECTIVE AMOUNT OF A COMPOUND OF FORMULA I.
来源网站:
中国工程科技知识中心
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