METASTIN DERIVATIVES AND ITS USE.

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专利权人:

TAKEDA PHARMACEUTICAL COMPANY LIMITED

发明人:

ASAMI, TAIJI,NISHIZAWA, NAOKI

申请号：

ES06843555

公开号：

ES2375038T3

申请日:

2006.12.21

申请国别(地区):

ES

年份:

2012

代理人:

摘要：

A metastine derivative selected from: Ac-D-Tyr-Aze (2) -Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 720), Ac-D-Tyr-Pic (2) -Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 721), Ac-D-Tyr-Hyp-Asn-Thr-Fe-AzaGly-Leu-Arg (5 Me) -Trp-NH2 (Compound No. 723), Ac-D-Tyr-Gly-Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 726), Ac-D- Tyr-Aib-Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 727), Ac-D-Tyr-D-NMeAla-Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 732), Ac-D-Tyr-Izc-Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 734), Ac-D -Tyr-D-Gln-Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 738), Ac-D-Tyr-D-His-Asn-Thr-Fe-AzaGly- Leu-Arg (Me) -Trp-NH2 (Compound No. 739), Ac-D-Tyr-Ala-Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 742), Ac-D-Tyr-Ser-Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 744), Ac-D-Tyr-Lys-Asn-Thr-Fe-AzaGly-Leu -Arg (Me) -Trp-NH2 (Compound No. 745), Ac-D-Tyr-Glu-Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 746), Ac -D- Tyr-D-Trp-Asn-Thr-Fe (3F) -AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 750), Ac-D-Tyr-Glu-Asn-Thr-Fe (2F) -AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 755), Ac-D-Tyr-Lys-Asn-Thr-Fe (3F) -AzaGly-Leu-Arg (Me) -Trp-NH2 ( Compound No. 756), Ac-D-Tyr-Glu-Asn-Thr-Fe (3F) -AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 757), Ac-D-Tyr-Lys- Asn-Thr-Fe (4Cl) -AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 758), Ac-D-Tyr-Glu-Asn-Thr-Fe (4Cl) -AzaGly-Leu-Arg (Me) -Trp-NHz (Compound No. 759), Ac-D-Tyr-Hyp-Asn-Thr-Fe (2F) -AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 763), Ac-D-Tyr-Hyp-Asn-Thr-Fe (3F) -AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 765), Ac-D-Tyr-Hyp-Asn-Thr-Fe ( 4Cl) -AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 767), Ac-D-Tyr-His (3Me) -Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp- NH2 (Compound No. 773), Ac-D-Tyr-Tyr (PO3H2) -Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 775), Glycoloil-D-Tyr- Hyp-Asn-Thr-Fe-AzaGly-Leu-Arg (Me) -Trp-NH2 (Compound No. 776), Ac-D-Tyr-Hyp-Asn-Thr-Fe

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