ARNE DR. SCHOLZ,ULF DR. BMER,PHILIP DR. LIENAU,GERHARD DR. SIEMEISTER,DIRK DR. KOSEMUND,ROLF DR. BOHLMANN,ULRICH DR. LCKING,NIELS DR. BHNKE
申请号：
ARP130104209
公开号：
AR093503A1
申请日:
2013.11.15
申请国别(地区):
AR
年份:
2015
代理人:
摘要：
Claim 1: a compound of General formula (1) where r u00b9 represents a group selected from c u2081 u208b u2086 c u2083 u208b u2087 alkyl, cycloalkyl, heterociclilo, phenyl heteroaryl alkyl, phenyl or heteroaryl alkyl c u2081 u208b u2083 c u2081 u208b u2083, where the group is optionally substituted with a Or two or three substituents, identically or differently, selected from the group consisting of Hydroxy Ciano,Halogen, alkoxy c u2081 u208b u2086 c u2081 u208b u2083 Halo alkyl, alkoxy, fluoro - c u2081 u208b u2083, nh u2082, alquilamino, dialquilamino, Acetylamino, N - methyl - N - acetylamino, cyclic amines, op (OR) (OH) u2082, - C (o) Oh, - C (o) nh u2082； R u00b2 represents a group selected among the Group of formulas (2)； r u00b3, r u2074 represent Independently, a group selected from a hydrogen Atom, an atom of Fluorine, Chlorine Atom,Bromine Atom, c u2081 u208b u2083 Ciano, alkyl, alkoxy c u2081 u208b u2083, Halo c u2081 u208b u2083 fluoro alkyl, alkoxy c u2081 u208b u2083； r u2075 represents a group selected from a hydrogen Atom, cyano, - C (o) r u2079, - C (o) - S (o) or u2079, u2082r u2079, - C (o) - nr u00b9 u2070r u00b9 u00b9, P (o) (or u00b9 u00b2) u2082, - ch u2082op (or u00b9 u00b2) u2082, alkyl c u2081 u208b u2086 c u2083 u208b u2087, cycloalkyl, heterociclilo, phenyl heteroaryl, where the alkyl group c u2081 u208b u2086 c u2083 u208b u2087, cycloalkyl, heterociclilo,PHENYL or heteroaryl is optionally substituted with one, two or three substituents, identically or differently selected from Halogen, Hydroxy, alkoxy alkyl, cyano, c u2081 u208b u2083, c u2081 u208b u2083, - nh u2082, alquilamino, dialquilamino, Acetylamino, N - methyl - N - acetylamino, cyclic amines, Hal C u2081 u208b u2083 fluoro alkyl or alkoxy, c u2081 u208b u2083； r u2076, r u2077 represent, independently,A group selected from a hydrogen Atom, an atom of Fluorine, Chlorine Atom, c u2081 u208b u2083 alkyl, alkoxy c u2081 u208b u2083, Halo c u2081 u208b u2083 fluoro alkyl, alkox
