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intermediates useful for the synthesis of a selective inhibitor against protein kinase and processes for preparing them
专利权人:
YUHAN CORPORATION
发明人:
DOO-BYUNG LEE,HYUN JU,JA-HEOUK KHOO,JONG-CHUL LIM,JUN-SUP LEE,JUNG-AE LEE,SANG-HO OH,SANG-SEOL JEON,WOO-SEOB SHIN
申请号:
BR112020001457
公开号:
BR112020001457A2
申请日:
2018.07.25
申请国别(地区):
BR
年份:
2020
代理人:
摘要:
the present invention relates to intermediates useful for the synthesis of an aminopyrimidine derivative or a pharmaceutically acceptable salt thereof having a selective inhibitory activity against protein kinases, especially against protein kinases for mutant epidermal growth factor receptors; and processes for preparing them. and the present invention also relates to intermediates useful for said process and processes for preparing them.a presente invenção refere-se a intermediários úteis para a síntese de um derivado de aminopirimidina ou um sal farmaceuticamente aceitável do mesmo tendo uma atividade inibidora seletiva contra proteínas quinases, especialmente contra proteínas quinases para receptores mutantes de fator de crescimento epidérmico; e processos para preparar os mesmos. e a presente invenção refere-se também a intermediários úteis para o dito processo e processos para preparar os mesmos.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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