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CRYSTALLINE FORM OF (R)-4-(5-(CYCLOPROPYLETHYNYL)ISOXAZOL-3-YL)-N-HYDROXY-2-METHYL-2-(METHYLSULFONYL)BUTANAMIDE AS AN ANTIBACTERIAL AGENT
专利权人:
NOVARTIS AG
发明人:
FU, Jiping,JIANG, Siyi,KORDIKOWSKI, Andreas,SWEENEY, Zachary Kevin
申请号:
SG11201810656W
公开号:
SG11201810656WA
申请日:
2017.06.12
申请国别(地区):
SG
年份:
2018
代理人:
摘要:
INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (43) International Publication Date 21 December 2017 (21.12.2017) WIP0 I PCT 0111111010 0111 inn Oil ioo monliflo oimIE (10) International Publication Number WO 2017/216705 Al (51) International Patent Classification: C07D 261/08 (2006.01) A61P 31/04 (2006.01) A61K 31/42 (2006.01) (21) International Application Number: PCT/IB2017/053468 (22) International Filing Date: 12 June 2017 (12.06.2017) (25) Filing Language: English (26) Publication Language: English (30) Priority Data: PCT/CN2016/085694 14 June 2016 (14.06.2016) CN (71) Applicant: NOVARTIS AG [CH/CH] Lichtstrasse 35, 4056 Basel (CH). (72) Inventors: FU, Jiping Novartis Institutes for BioMedical Research Inc., 5300 Chiron Way, Emeryville, California 94608 (US). JIANG, Siyi Beijing Novartis Pharma Co. Ltd., 4218 Jinke Road, Zhangjiang Hi-Tech Park, Shang- hai 201203 (CN). KORDIKOWSKI, Andreas Novartis Pharma AG, Postfach, CH-4002 Basel (CH). SWEENEY, Zachary Kevin 143 King Street, Redwood City, Califor- nia 94602 (US). (74) Agent: NOVARTIS AG Lichtstrasse 35, 4056 Basel (CH). (81) Designated States (unless otherwise indicated, for every kind of national protection available): AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW. (84) Designated States (unless otherwise indicated, for every kind of regional protection available): ARIPO (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW), Eurasian (AM, AZ, BY, KG, KZ, RU, TJ, T
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/
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