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SALT FORMS OF 4-(4-METHYLPIPERAZIN-1-YLMETHYL)-n-[4-METHYL-3-(4-PYRIDIN-3-YL)PYRIMIDIN-2-YLAMINO)PHENYL]-BENZAMIDE
专利权人:
NOVARTIS AG
发明人:
HANS MICHAEL BURGER,PAUL WILLIAM MANLEY,MICHAEL MUTZ
申请号:
PH12013500157
公开号:
PH12013500157A1
申请日:
2013.01.22
申请国别(地区):
PH
年份:
2014
代理人:
摘要:
The present invention relates to acid addition salts of 4-[4-methyl-1-piperazinylmethyl]-N-[4-methyl-3-[[4-3-pyridinyl-2-pyrimidinyl]amino]phenyl]-benzamide, which are selected from the group consisting of a tartrate salt, such as a (D)(-) tartrate salt or a (L)(+) tartrate salt, a hydrochloride salt, a citrate sat, a malate salt, a fumarate salt, a succinate salt, a benzoate salt, a benzenesulfonate salt, a pamoate salt, a formate salt, a malonate salt, a 1,5-naphthalenedisulfonate salt, a salicylate salt, a cyclohexanesulfamate salt, a lactate salt, a mandelate salt, aq glutarate salt, an adipate salt, a squarate salt, a vanillate salt, an oxaloacetate salt, an ascorbate salt and a sulfate salt.
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