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alkynyl-derived compounds as metabotropic glutamate receptor modulators, their uses and their pharmaceutical compositions
专利权人:
ADDEX PHARMACEUTICALS SA;ADDEX PHARMA S.A.
发明人:
Anne-Sophie Bessis,Béatrice Bonnet,Christelle Bolea,Jean-Philippe Rocher,Mark Epping-Jordan,Nicholas Poirier,Sonia-Maria Poli,Yves Thollon
申请号:
BRPI0511072
公开号:
BRPI0511072B1
申请日:
2005.06.17
申请国别(地区):
BR
年份:
2019
代理人:
摘要:
alkynyl derivatives as metabotropic glutamate receptor modulators. The present invention relates to novel compounds of formula (I) wherein w, n, x and w? are defined in the description; The compounds of the invention are modulators of the metabotropic glutamate receptor subtype 5 ("mgiur5") which are useful for treating central nervous system disorders as well as other m-giur5 receptor modulated disorders.derivados de alquinila como moduladores dos receptores de glutamato metabotróbico.a presente invenção refere-se a novos compostos de fórmula (i) em que w, n, x e w<;39>; são definidos na descrição; os compostos da invenção são moduladores dos receptores de glutamato metabotrópico - subtipo 5 ("mgiur5") que são úteis para o tratamento de distúrbios do sistema nervoso central assim como outros distúrbios modulados pelos receptores de m-giur5.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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