您的位置: 首页 > 农业专利 > 详情页

PROCESS FOR THE PREPARATION OF BENZOIMIDAZOL-2-YL PYRIMIDINE DERIVATIVES
专利权人:
JANSSEN PHARMACEUTICA N.V.
发明人:
CESCO-CANCIAN, SERGIO,GRIMM, JEFFREY, S,MANI, NEELAKANDHA, S,MAPES, CHRISTOPHER, M,PALMER, DAVID, C,PIPPEL, DANIEL, J,XIAO, TONG,BROGGINI, DIEGO,LOCHNER, SUSANNE
申请号:
NZ59016909
公开号:
NZ590169A
申请日:
2009.06.29
申请国别(地区):
NZ
年份:
2012
代理人:
摘要:
Disclosed herein is a process for the preparation of a compound of formula (I) and derivatives (I-A) and (I-B), wherein the substituents are as defined within the specification, comprising the steps of: reacting a compound of formula (V) with a reducing agent system; in a solvent; at a temperature in the range of from about 0°C to 25°C, to yield a compound of formula (VI); followed by reacting a compound of formula (VI) with a compound of formula (VII) in the presence of an oxidizing agent system, in a solvent, at a temperature in the range of from about 20°C to 100°C to afford the compound of formula (I).
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

意 见 箱

匿名:登录

个人用户登录

找回密码

第三方账号登录

忘记密码

个人用户注册

必须为有效邮箱
6~16位数字与字母组合
6~16位数字与字母组合
请输入正确的手机号码

信息补充