Dipicolylamine compounds of Formula (I) set forth herein. Also disclosed are pharmaceutical compositions containing metal ions and these compounds. Further disclosed is a method for treating a condition associated with cells containing inside-out phosphatidylserine, with these compounds.本發明係提供一種式(I)之二甲基吡啶胺化合物,另提供一種包含金屬離子和這類化合物之醫藥組成物,再提供一種使用這類化合物治療與含磷脂質絲胺酸進出之細胞相關病症之方法。