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Macrocycles as Kinase Inhibitors
- 专利权人:
- MERCK PATENT GESELLSCHAFT MIT BESCHRÄNKTER HAFTUNG
- 发明人:
- GUENTER DR. HOELZEMANN,DIETER DR. DORSCH,ANSGAR DR. WEGENER,OLIVER DR. POESCHKE,MICHAEL DR. BUSCH
- 申请号：
- ARP140101780
- 公开号：
- AR096149A1
- 申请日:
- 2014.04.30
- 申请国别(地区):
- AR
- 年份:
- 2015
- 代理人:
- 摘要：
- Claim 1: compounds of the formula (1) where X denotes N or CH and denotes het dilaurate or AR q\u00b9 denotes \u2099 (ch\u2082), or (ch\u2082) or \u2099 (ch\u2082 \u2099het\u00b9 - di\u00edlo) (m denotes \u209anr\u00b3co, conr\u00b3, ch\u2082)Nr\u00b3 or co q\u00b2 denotes (ch\u2082) \u2099o \u2099 or (b ch\u2082) denotes ar or het het denotes dilaurate Furan, thiophene, pyrrole, imidazole, pyrazole, oxazole, isoxazole, triazole, Oxadiazoles, thiazole, pyridine, pyrimidine, tetrazol,Pyridazine hydrochloride, pyrazine, isoindolindolina, indole, quinoline, isoquinoline indazol, benzimidazole, benzoxazole, 1.3 - benzo dioxol, benzothiophene, benzofuran, imidazopiridina, dihidroindol, quinoxaline,Benzo [1,2,5] thiadiazole or furo [3,2-b] pyridine, each of which is not replaced or mono - or alkylated with Hal, (r\u00b3) \u2082 [c] \u209aor\u00b3 [c] (r\u00b3) \u2082 \u209an (r\u00b3) \u2082 [c] \u209ahet\u00b9 \u2082 (r\u00b3), no\u2082, CN, (\u2082 [c] \u209acoor\u00b3, r\u00b3)With \u2082 (r\u00b3), nr\u00b3coa, nr\u00b3so\u2082a, so\u2082n (\u2082 r\u00b3), S (OR) \u2099a cohet\u00b9,, or [C (r\u00b3) \u2082 \u2098n (r\u00b3) \u2082], or [c] (r\u00b3) \u2082 \u209ahet\u00b9, nhcooa, nhcon (r\u00b3) \u2082, nhcoo [c] \u2082 (r\u00b3) \u2098n (r\u00b3), nhcoo [c] (r\u00b3) \u2082 \u209ahet\u00b9, nhconh [c] (r\u00b3) \u2082 \u2098n (r\u00b3) \u2082, nhconh [c] \u209ahet\u00b9 \u2082 (r\u00b3),Oconh [c] (r\u00b3) \u2082 \u2098n (r\u00b3) \u2082, oconh [c] (r\u00b3) \u2082 \u209ahet\u00b9, Cho, coa = S = U = nr\u00b3 and \/ or sulfide ar denotes, that is not replaced or is mono -, di - or trisustituido with Hal, [C (r\u00b3) \u209aor\u00b3 \u2082], or [c] \u209aor\u00b3 \u2082 (r\u00b3),[c] (r\u00b3) \u2082 \u209an (r\u00b3) \u2082 or [c] (r\u00b3) \u2082 \u209an (r\u00b3) \u2082 [c] (r\u00b3) \u2082 \u209ahet\u00b9, no\u2082, CN, [C (r\u00b3) \u209acoor\u00b3 \u2082], or [c] \u209acoor\u00b3 \u2082 (r\u00b3), with \u2082 (r\u00b3) nr\u00b3coa nr\u00b3so\u2082a (,,, so\u2
- 来源网站：
- 中国工程科技知识中心
- 来源网址：
- http://www.ckcest.cn/home/
