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PROCESS FOR THE PREPARATION OF GLUCURONIDE DRUG-LINKERS AND INTERMEDIATES THEREOF
专利权人:
INC.;SEATTLE GENETICS
发明人:
MAO, Yunyu,MOQUIST, Philip,CHOUDHURY, Anusuya,DOUBLEDAY, Wendel
申请号:
SG11201908325P
公开号:
SG11201908325PA
申请日:
2018.03.23
申请国别(地区):
SG
年份:
2019
代理人:
摘要:
INTERNATIONAL APPLICATION PUBLISHED UNDER THE PATENT COOPERATION TREATY (PCT) (19) World Intellectual Property Organization International Bureau (43) International Publication Date 27 September 2018 (27.09.2018) WIPO I PCT ill 1111u°11111VIIIVIIII o oloincioimommo oimIE (10) International Publication Number WO 2018/175994 Al (51) International Patent Classification: A61K 47/64 (2017.01) C07H 15/203 (2006.01) A61K 47/68 (2017.01) (21) International Application Number: PCT/US2018/024191 (22) International Filing Date: 23 March 2018 (23.03.2018) (25) Filing Language: English (26) Publication Language: English (30) Priority Data: 62/476,605 24 March 2017 (24.03.2017) US (71) Applicant: SEATTLE GENETICS, INC. [US/US]; 21823 30th Drive SE, Bothell, Washington 98021 (US). (72) Inventors: MAO, Yunyu; 21823 30th Drive SE, Both- ell, Washington 98021 (US). MOQUIST, Philip; 21823 30th Drive SE, Bothell, Washington 98021 (US). CHOUD- HURY, Anusuya; 21823 30th Drive SE, Bothell, Washing- ton 98021 (US). DOUBLEDAY, Wendel; 21823 30th Dri- ve SE, Bothell, Washington 98021 (US). (74) Agent: CASTELLINO, Angelo et al.; Seattle Genetics, INC., 21823 30TH Drive SE, Bothell, Washington 98021 (US). = (81) Designated States (unless otherwise indicated, for every kind of national protection available): AE, AG, AL, AM, AO, AT, AU, AZ, BA, BB, BG, BH, BN, BR, BW, BY, BZ, CA, CH, CL, CN, CO, CR, CU, CZ, DE, DJ, DK, DM, DO, DZ, EC, EE, EG, ES, FI, GB, GD, GE, GH, GM, GT, HN, HR, HU, ID, IL, IN, IR, IS, JO, JP, KE, KG, KH, KN, KP, KR, KW, KZ, LA, LC, LK, LR, LS, LU, LY, MA, MD, ME, MG, MK, MN, MW, MX, MY, MZ, NA, NG, NI, NO, NZ, OM, PA, PE, PG, PH, PL, PT, QA, RO, RS, RU, RW, SA, SC, SD, SE, SG, SK, SL, SM, ST, SV, SY, TH, TJ, TM, TN, TR, TT, TZ, UA, UG, US, UZ, VC, VN, ZA, ZM, ZW. (84) Designated States (unless otherwise indicated, for every kind of regional protection available): ARIPO (BW, GH, GM, KE, LR, LS, MW, MZ, NA, RW, SD, SL, ST, SZ, TZ, UG, ZM, ZW), Eurasian (AM, AZ, BY, KG, KZ, RU,
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