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CYCLOPROPANE COMPOUNDS
专利权人:
EISAI R&D MANAGEMENT CO.; LTD.
发明人:
TERAUCHI TARO,TAKEMURA AYUMI,DOKO TAKASHI,YOSHIDA YU,TANAKA TOSHIAKI,SORIMACHI KEIICHI,NAOE YOSHIMITSU,BEUCKMANN CARSTEN,KAZUTA YUJI
申请号:
MYPI 2013000954
公开号:
MY160969A
申请日:
2011.09.20
申请国别(地区):
MY
年份:
2017
代理人:
摘要:
A CYCLOPROPANE COMPOUND REPRESENTED BY THE FOLLOWING FORMULA (A) OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF HAS OREXIN RECEPTOR ANTAGONISM, AND THEREFORE HAS A POTENTIAL OF USEFULNESS FOR THE TREATMENT OF SLEEP DISORDER FOR WHICH OREXIN RECEPTOR ANTAGONISM IS EFFECTIVE, FOR EXAMPLE, INSOMNIA: WHEREIN Q REPRESENTS -CH- OR A NITROGEN ATOM, R1A AND R1B EACH INDEPENDENTLY REPRESENT A C1-6 AIKYL GROUP AND THE LIKE, R1C REPRESENTS A HYDROGEN ATOM AND THE LIKE, R2A, R2B, R2C AND R2D EACH INDEPENDENTLY REPRESENT A HYDROGEN ATOM, A HALOGEN ATOM, A C1-6 ALKYL GROUP AND THE LIKE, R3A, R3B AND R3C EACH INDEPENDENTLY REPRESENT A HYDROGEN ATOM, A HALOGEN ATOM AND THE LIKE, AND R3D REPRESENTS A HYDROGEN ATOM AND THE LIKE. (FIGURE 1)
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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