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PROCESS FOR PREPARING TIANEPTIN AND ITS PHARMACEUTICALLY ACCEPTABLE SALTS AND 11-AMINO-3-CHLORINE 6,11-DIIDRO-5,5-DIOXO-6-METHYL-DIBENZO [c, f] [1,2] -TAZAZINE
专利权人:
LES LABORATOIRES SERVIER
发明人:
JACKY BLANCHARD,HUGUES TURBE,DANIEL BRIGOT
申请号:
BR0101230
公开号:
BR0101230B1
申请日:
2001.03.29
申请国别(地区):
BR
年份:
2013
代理人:
摘要:
Synthesis of 11-amino-3-chloro-6,11-dihydro-5,5-dioxo-6-methyl dibenzo(c,f)(1,2)thiazepine (I) and its salts, from 3-chloro-6,11-dihydro-6-methyl-5,5,11-trioxo dibenzo(c,f)(1,2)thiazepine (III). Synthesis of 11-amino-3-chloro-6,11-dihydro-5,5-dioxo-6-methyl dibenzo(c,f)(1,2)thiazepine of formula (I) and its salts, from 3-chloro-6,11-dihydro-6-methyl-5,5,11-trioxo dibenzo(c,f)(1,2)thiazepine of formula (III): Independent claims are also included for the use of (I) to prepare tianeptine (II) and its salts.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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