Mahesh Khedekar;Sukumar Sinha;Mubeen Ahmed Khan;Ramjilal Yadav;Navin Ganesh Bhatt;Nikhil Rasiklal Trivedi
发明人:
Navin Ganesh Bhatt,Nikhil Rasiklal Trivedi,Mahesh Khedekar,Sukumar Sinha,Mubeen Ahmed Khan,Ramjilal Yadav
申请号：
US13003885
公开号：
US08623844B2
申请日:
2009.07.17
申请国别(地区):
US
年份:
2014
代理人:
摘要：
The present invention generally relates to a process for the preparation of fosaprepitant dimeglumine intermediate and its use in the preparation of fosaprepitant dimeglumine； to a neutral form of fosaprepitant in a solid state and processes for the preparation thereof； and to a stable amorphous fosaprepitant dimeglumine, having a stability at temperatures of about 2° C. to about 8° C. and at a relative humidity below at least 60%； and a process for the preparation thereof.
