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COMPOUND OR SALT OF THE SAME, PRODUCT, PHARMACEUTICAL AGENT, METHODS FOR ANTAGONIZING AN ANDROGEN RECEIVER AND FOR PREVENTING / TREATING CANCER, AND, USE OF THE COMPOUND OR PRODUCT OF THE SAME.
专利权人:
TAKEDA PHARMACEUTICAL COMPANY LIMITED
发明人:
MITSUHIRO ITO,TOMOHIKO SUZAKI,SATOSHI YAMAMOTO
申请号:
BRPI0816095
公开号:
BRPI0816095A2
申请日:
2008.08.27
申请国别(地区):
BR
年份:
2015
代理人:
摘要:
The present invention provides a novel pyrazole derivative and an androgen receptor antagonist containing the derivative. The present invention provides a compound represented by the formula (I') wherein R 1 is a hydrogen atom, a group via a carbon atom, a group via a nitrogen atom, a group via an oxygen atom, or a group via a sulfur atom; R 2 is a phenyl group having cyano (the phenyl group may further have substituent(s) other than cyano); R 3 is a hydrogen atom, a group via a carbon atom, a group via a nitrogen atom, a group via an oxygen atom, or a group via a sulfur atom; R 4 is a cyclic group optionally having substituent(s); and X is methylene optionally having substituent(s), or CO, or a salt thereof.
来源网站:
中国工程科技知识中心
来源网址:
http://www.ckcest.cn/home/

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