WÜNSCH, BERNHARD,SCHEPMANN, DIRK,SCHLÄGER, TORSTEN,ZAMANILLO-CASTANEDO, DANIEL
申请号：
ES08748940
公开号：
ES2472741T3
申请日:
2008.04.16
申请国别(地区):
ES
年份:
2014
代理人:
摘要：
A compound of general formula Ia, ** Formula ** in which p is selected from 0 or 1； R1 is selected from linear or branched C1-4 alkyl； or optionally at least monosubstituted aryl； R2 is selected from H； OH or a linear or branched C1-4 alkyl group； R3 is selected from hydrogen； C1-10 alkyl, linear or branched； C3-8 alkenyl, linear or branched； (C1-6) alkyl optionally at least monosubstituted aryl； (C1-6) alkyl optionally at least monosubstituted heterocyclyl； or (C1-6) alkyl (C4-8) cycloalkyl optionally at least monosubstituted, in which the cycloalkyl group may be saturated or unsaturated, optionally in the form of one of the stereoisomers, preferably enantiomers or diastereomers, a racemate or in the form of a mixture of at least two of the stereoisomers, preferably enantiomers and / or diastereomers, at any mixing rate, or a corresponding salt thereof, or a corresponding solvate thereof, in which the aryl or alkyl-aryl groups, cycloalkyl or alkyl-cycloalkyl, heterocyclyl or alkyl-heterocyclyl, are substituted in the aryl or alkyl-aryl, cycloalkyl or alkyl-cycloalkyl, heterocyclyl or alkylheterocyclyl ring system, by substituents selected from OH, SH,>； = O, halogen ( F, Cl, Br, I), CN, NO2, COOH； NRxRy, with Rx and Ry independently being H or a C1-6 alkyl saturated or unsaturated, linear or branched, substituted or unsubstituted； a saturated or unsaturated, linear or branched, substituted or unsubstituted -O-C 1-6 alkyl (alkoxy)； a -C1-6 saturated or unsaturated, linear or branched, substituted or unsubstituted； a -C (O) -C1-6 saturated or unsaturated, linear or branched, substituted or unsubstituted group； a -C (O) -O-C1-6 saturated or unsaturated, linear or branched, substituted or unsubstituted group； a substituted or unsubstituted aryl or alkyl-aryl； a substituted or unsubstituted cycloalkyl or alkylcycloalkyl； a substituted or unsubstituted heterocyclyl or alkyl heterocyclyl and in which alkyls or alkenyls may be substituted or unsubstituted, in which the a
