process for the preparation of a chiral compound, chiral compound, composition, pharmaceutical composition, use of a composition, method of treatment or prevention and use of a compound
DOMINIC DE SOUZA,HANS-PETER SPITZENSTÄTTER,HUBERT STURM,JÖRG SALCHENEGGER,MARTIN ALBERT,MARTIN LANGNER,MICHAEL OBERHUBER,THORSTEN WILHELM
申请号：
BR112012029227
公开号：
BR112012029227A2
申请日:
2011.05.18
申请国别(地区):
BR
年份:
2016
代理人:
摘要：
A process for the preparation of a chiral compound, in particular posaconazole, wherein the process comprises mixing and reacting the compounds of formula (I) Y3&mdash；NH2； of formula (IIa) 0=C&boxH；N&mdash；Y0 and/or of formula (IIb) and of formula (III) in a solvent in any order to obtain a reaction mixture containing a chiral compound of formula (IV) and/or formula (V).
