BUCHSTALLER, HANS-PETER,WIESNER, MATTHIAS,ZENKE, FRANK,AMENDT, CHRISTIANE,GRELL, MATTHIAS,SIRRENBERG, CHRISTIAN
申请号:
ES04739826
公开号:
ES2465624T3
申请日:
2004.06.11
申请国别(地区):
ES
年份:
2014
代理人:
摘要:
Benzimidazole carboxamides of the formula I ** Formula ** wherein R6, R7 are independently from each other H or AA is independently selected from the group consisting of alkyl, alkoxy and alkoxyalkyl, Ar2 is pyridinyl, R8 is selected from the group consisting of alkyl comprising 1 to 4 carbon atoms, alkoxy comprising 1 to 4 carbon atoms, Hal, CH2Hal, CH (Hal) 2, perhaloalkyl comprising 1 to 4 carbon atoms, NO2 and (CH2) nCN, R9 and R10 are independently selected from a group consisting of H, A, cycloalkyl comprising 3 to 7 carbon atoms, Hal, CH2Hal, CH (Hal) 2, C (Hal) 3, NO2, (CH2) nCN, (CH2) nNR11R12, (CH2) nOR11, (CH2) nO (CH2) kNR11R12, (CH2) nCOOR12, (CH2) nCONR11R12, (CH2) nNR11COR13, (CH2) nNR11CONR11R12, (CH2) nNR11SO2A, (CH2) nS2 (O) uR13, (CH2) nOC (O) R13, (CH2) nCOR13, (CH2) nSR11, CH>; = NOA, CH2CH>; = N-OA, (CH2) nNHOA, (CH2) nCH>; = N-R11 , (CH2) nOC (O) NR11R12, (CH2) nNR11COOR12, (CH2) nN (R11) CH2CH2OR13, (CH2) nN (R11) CH2CH2OCF3. (CH2) nN (R11) C (R13) HCOOR12, C (R13) HCOR12, (CH2) nN (R11) CH2CH2N (R12) CH2COOR12, (CH2) nN (R11) CH2CH2NR11R12, CH>; = CHCOOR11, CH>; = CHCH2NR11R12 , CH>; = CHCH2NR11R12, CH>; = CHCH2OR13, (CH2) nN (COOR11) COOR12, (CH2) nN (CONH2) COOR11, (CH2) nN (CONH2) CONH2, (CH2) nN (CH2COOR11) COOR12, (CH2) nN (CH2CONH2) COOR11, (CH2) nN (CH2CONH2) CONH2, (CH2) nCHR13COR11, (CH2) nCHR13COOR1120, (CH2) nCHR13CH2OR14, (CH2) nOCN and (CH2) nNCO.Benzimidazol carboxamidas de la fórmula I**Fórmula** en donde R6, R7 son independientemente uno de otro H o A A se selecciona independientemente del grupo que consiste en alquilo, alcoxi y alcoxialquilo, Ar2 es piridinilo, R8 se selecciona del grupo que consiste en alquilo que comprende de 1 a 4 átomos de carbono, alcoxi que comprende 1 a 4 átomos de carbono, Hal, CH2Hal, CH(Hal)2, perhaloalquilo que comprende 1 a 4 átomos de carbono, NO2 y (CH2)nCN, R9 y R10 se seleccionan independientemente de un grupo que consiste en H, A, cicloalquilo que comprende 3 a 7 átomos de carb