GOULET, MARK T.,NARGUND, RAVI P.,SEBHAT, IYASSU K.,UJJAINWALLA, FEROZE,WALSH, THOMAS F.,WARNER, DANIEL,YE, ZHIXIONG,YOUNG, JONATHAN R.,BAKSHI, RAMAN K.
申请号:
CA2439149
公开号:
CA2439149C
申请日:
2002.02.25
申请国别(地区):
CA
年份:
2012
代理人:
摘要:
Certain novel 4-substituted N-acylated piperidine derivatives of formula (I)areagonists of the human melanocortin receptor(s) and, in particular, areselective agonists of thehuman melanocortin-4 receptor (MC-4R). They are therefore useful for thetreatment,control, or prevention of diseases and disorders responsive to the activationof MC-4R, suchas obesity, diabetes, sexual dysfunction, including erectile dysfunction andfemale sexualdysfunction(see formula I)