The present application relates to novel (3-hydroxyphenyl)amino-substituted pyrido[2,3-b][1,5]benzodiazepin-5-one derivatives, to processes for preparation thereof, to the use thereof alone or in combination for treatment and/or prevention of diseases and to the use thereof for production of medicaments for treatment and/or prevention of diseases, especially of angiogenic disorders and hyperproliferative disorders in which neovascularization plays a role, for example ophthalmological disorders and cancers and tumours. Such treatments can be effected as monotherapy or else in combination with other medicaments or further therapeutic measures.本申請案係有關一種新穎之(3-羥苯基)胺基-取代之吡啶並[2,3-b][1,5]苯並二氮呯-5-酮衍生物、其製法、其於治療及/或預防疾病上之單獨用途或組合用途、及其於製造用於治療及/或預防疾病(尤指以新生血管為重要因素之生成血管性病變及過度增生性病變,例如:眼睛病變及癌症與腫瘤)之醫藥上之用途。此等治療法可依單方療法或與其他醫藥或其他醫療法組合進行。
