KIM, SOON-HOE,IM, WEON-BIN,CHOI, SUNG-HAK,CHOI, SUN-HO,SOHN, JU-HEE,SUNG, HYUN-JUNG,KIM, MI-YEON,CHO, KANG-HUN,SOHN, TAE-KYOUNG
申请号:
MYPI 2012004698
公开号:
MY162554A
申请日:
2011.04.18
申请国别(地区):
MY
年份:
2017
代理人:
摘要:
THE PRESENT INVENTION PROVIDES A NOVEL BENZAMIDE DERIVATIVE OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF, A METHOD FOR PREPARING THE SAME, AND A 5-HT4 RECEPTOR AGONIST CONTAINING THE SAME AS AN ACTIVE INGREDIENT. BENZAMIDE DERIVATIVES OF THE PRESENT INVENTION HAVE A SUPERIOR AFFINITY FOR 5-HT4 RECEPTORS, A CAPABILITY TO REDUCE A GASTRIC EMPTYING TIME AND A LOW TOXICITY, AND CONSEQUENTLY ARE THERAPEUTICALLY EFFECTIVE FOR THE TREATMENT OF A VARIETY OF DISEASES ASSOCIATED WITH 5-HT4 RECEPTORS.