Robert James Pasteris;Rafael Shapiro;Mary Ann Hanagan;Matthew Richard Oberholzer
发明人:
Mary Ann Hanagan,Matthew Richard Oberholzer,Robert James Pasteris,Rafael Shapiro
申请号：
US13265138
公开号：
US20120034315A1
申请日:
2010.04.19
申请国别(地区):
US
年份:
2012
代理人:
摘要：
Disclosed are solid forms of 1-[4-[4-[5-(2,6-difluorophenyl)-4,5-dihydro-3-isoxazolyl]-2-thiazolyl]-1-piperidinyl]-2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethanone (Compound 1). Methods for the preparation of solid forms of Compound 1 and for the conversion of one solid form of Compound 1 into another are disclosed.Disclosed are fungicidal compositions comprising a fungicidally effective amount of a solid form of Compound 1 and at least one additional component selected from the group consisting of surfactants, solid diluents and liquid carriers. Compositions comprising a mixture of a solid form of Compound 1 and at least one other fungicide or insecticide are also disclosed.Also disclosed are methods for controlling plant diseases caused by fungal plant pathogens comprising applying to a plant or portion thereof, or to a plant seed, a fungicidally effective amount of a solid form of Compound 1.
